2019 – 2020
81. Synthesis and Structure–Activity Relationship of Dehydrodieugenol B Neolignans against Trypanosoma cruzi
C. E. Sear, P. Pieper, M. Amaral, M. M. Romanelli, T. A. Costa-Silva, M. M. Haugland, J. A. Tate, J. H. G. Lago, A. G. Tempone*, E. A. Anderson*
ACS Infect. Dis., 2020, doi: 10.1021/acsinfecdis.0c00523
80. Site-Selective C–H Benzylation of Alkanes with N-Triftosylhydrazones Leading to Alkyl Aromatics
Z. Liu, S. Cao, W. Yu, J. Wu, F. Yi, E. A. Anderson*, X. Bi*
Chem, 2020, 6, 2110–2124, doi: 10.1016/j.chempr.2020.06.031
79. Copper-Catalyzed Intramolecular C–H Alkoxylation of Diaryltriazoles: Synthesis of Tricyclic Triazole Benzoxazines
X. Ma, H. Li, H. Xin, W. Du, E. A. Anderson*, X. Dong*, Y. Jiang*
Org. Lett., 2020, 22, 5320–5325 doi: 10.1021/acs.orglett.0c01517
78. Structure-activity relationship study of cytotoxic neolignan derivatives using multivariate analysis and computation-aided drug design
F. S. de Sousa, J. L. Baldim, R. A. Azevedo, C. R. Figueiredo, P. Pieper,
C. E. Sear, E. A. Anderson, J. H. G. Lago
Bioorg. Med. Chem. Lett., 2020, 30, 127349,
doi: 10.1016/j.bmcl.2020.127349
77. Synthesis of All-carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron-Catalyzed Kumada Cross-Coupling
J. Nugent,‡ B. R. Shire,‡, D. F. J. Caputo, H. D. Pickford, F. Nightingale,
I. T. T. Houlsby, J. J. Mousseau, E. A. Anderson
‡equal author contribution
Article: Angew. Chem. Int. Ed., 2020, 59, 11866–11870,
doi: 10.1002/anie.202004090
Featured in: Org. Process Res. Dev., 2020, doi: 10.1021/acs.oprd.0c00344
76. Rationalizing the diverse reactivity of [1.1.1]propellane through 𝜎-𝜋-delocalization
A. J. Sterling, A. B. Dürr, R. C. Smith, E. A. Anderson, F. Duarte
Chem. Sci., 2020, 11, 4895–4903. doi: 10.1039/D0SC01386B
75. 2′-Alkynyl spin-labelling is a minimally perturbing tool for DNA structural analysis
J. S. Hardwick, M. M. Haugland, A. H. El-Sagheer, D. Ptchelkine,
F. R. Beierlein, A. N. Lane, T. Brown, J. E. Lovett, E. A. Anderson
Nucleic Acids Research, 2020, 48, 2830–2840. doi: 10.1093/nar/gkaa086
74. A Modular, Enantioselective Synthesis of Resolvins D3, E1, and Hybrids
F. Urbitsch, B. L. Elbert, J. Llaveria, P. E. Streatfeild, E. A. Anderson
Org. Lett., 2020, 22, 1510–1515. doi: 10.1021/acs.orglett.0c00089
73. Enantioselective synthesis and anti-parasitic properties of aporphine natural products
P. Pieper, E. McHugh, M. Amaral, A. G.Tempone, E. A.Anderson
Tetrahedron., 2019, 76, 130814. doi: 10.1016/j.tet.2019.130814
72. Synthesis of Cyclic Alkenyl Dimethylsiloxanes from Alkynyl Benzyldimethylsilanes and Application in Polyene Synthesis
H. G. Gudmundsson, C. J. Kuper, D. Cornut, F. Urbitsch, B. L. Elbert,
E. A. Anderson
J. Org. Chem., 2019, 84, 14868-14882. doi: 10.1021/acs.joc.9b01664
71. Convergent Total Syntheses of (–)-Rubriflordilactone B and (–)-pseudo-Rubriflordilactone B
M. Mohammad, V. Chintalapudi, J. M. Carney, S. J. Mansfield, P. Sanderson, K. E. Christensen, E. A. Anderson
Angew. Chem. Int. Ed., 2019, 58, 18177–18181.
doi: 10.1002/anie.201908917
70. Dehydrodieugenol B derivatives as antiparasitic agents: Synthesis and biological activity against Trypanosoma cruzi
D. D. Ferreira, F. S. Sousa, T. A. Costa-Silva, J. Q. Reimão, A. C. Torrecilhas, D. M. Johns, C. E. Sear, K. M. Honorio, J. H. G. Lago, E. A. Anderson, A. G. Tempone
Eur. J. Med. Chem., 2019, 176, 162-174. doi: 10.1016/j.ejmech.2019.05.001
69. A semi-synthetic neolignan derivative from dihydrodieugenol B selectively affects the bioenergetic system of Leishmania infantum and inhibits cell division
M. Amaral, F. S. de Sousa, T. A. Costa Silva, A. Jimenez G. Junior, N. N. Taniwaki, D. M. Johns, J. H. G. Lago, E. A. Anderson & A. G. Tempone
Scientific Reports, 2019, 6, 6114. doi: 10.1038/s41598-019-42273-z
68. Silver-Catalyzed C- to N-Center Remote Arene Migration
Y. Ning, A. Mekareeya, K. R. Babu, E. A. Anderson and X. Bi
ACS Catalysis, 2019, 9, 4203-4210. doi: 10.1021/acscatal.9b00500
67. A General Route to Bicyclo[1.1.1]pentanes through Photoredox Catalysis.
J. Nugent,* C. Arroniz,* B. R. Shire, A. J. Sterling, H. D. Pickford, M. L. J. Wong, S. J. Mansfield, D. F. J. Caputo, B. Owen, J. J. Mousseau, F. Duarte and E. A. Anderson
*equal author contribution
ACS Catalysis, 2019, 9, 9568-9574. doi: 10.1021/acscatal.9b03190
66. A General Copper-Catalyzed Synthesis of Ynamides from 1,2-Dichloroenamides.
S. J. Mansfield, R. C. Smith, J. R. J. Yong, O. L. Garry, and E. A. Anderson
Org. Lett., 2019, 21, 2918-2922. doi: 10.1021/acs.orglett.9b00971.
65. Synthesis of Enantioenriched α-Chiral Bicyclo[1.1.1]pentanes.
M. L. J. Wong, J. J. Mousseau, S. J. Mansfield and E. A. Anderson.
Org. Lett., 2019, 21, 2408-2411. doi: 10.1021/acs.orglett.9b00691.
64. Palladium-catalysed ligand-free reductive Heck cycloisomerisation of 1,6-en-α-chloro-enamides.
Y. Hou, J. Ma, H. Yang, E. A. Anderson, A. Whiting and N. Wu.
Chem. Commun., 2019, 55, 3733-3736. doi: 10.1039/C9CC00537D.
63. Direct Transformation of Terminal Alkynes into Amidines by a Silver-Catalyzed Four-Component Reaction.
B. Liu, Y. Ning, M. Virelli, G. Zanoni, E. A. Anderson and X. Bi.
J. Am. Chem. Soc., 2019, 141, 1593-1598. doi: 10.1021/jacs.8b11039.
62. Use of trifluoroacetaldehyde N-tfsylhydrazone as a trifluorodiazoethane surrogate and its synthetic applications.
X. Zhang, Z. Liu, X. Yang, Y. Dong, M. Virelli, G. Zanoni, E. A. Anderson and X. Bi.
Nature Commun., 2019, 10, 284. doi: 10.1038/s41467-018-08253-z.
