2019 – 2021
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91. Synthesis of the C1–C27 Fragment of Stambomycin D Validates Modular Polyketide Synthase-Based Stereochemical Assignments

 

J. Lim,‡ V. Chintalapudi,‡ H.G. Gudmundsson, M. Tran, A. Bernasconi, A. Blanco, L. Song, G.L. Challis, and E.A. Anderson*

 

Org. Lett.2021, ASAP Article, 

doi: https://doi.org/10.1021/acs.orglett.1c02650

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90. Regio- and stereoselective addition of Brønsted acids to yndiamides: Synthesis of N,O,N- and N,S,N-trisubstituted ketene acetals

 

O.L Garry, S.J. Mansfield, and E.A. Anderson*

 

Synthesis2021, accepted, doi: https://doi.org/10.1055/a-1638-5783

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89. Synthesis of Polysubstituted Fused Pyrroles by Gold-Catalyzed Cycloisomerization/1,2-Sulfonyl Migration of Yndiamides

 

P.J. Smith, Y. Jiang, Z. Tong, H.D. Pickford, K.E. Christensen, J. Nugent, and E.A. Anderson*

 

Org. Lett.2021, 23, 6547–6552,

doi: https://doi.org/10.1021/acs.orglett.1c02360

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88. Recent progress in the total synthesis of pyrrole-containing natural products (2011–2020)

 

N. Singh,‡ S. Singh,‡ S. Kohli, A. Singh, H. Asiki, G. Rathee, R. Chandra,* and E.A. Anderson*

 

Org. Chem. Front.2021, Advance Article,

doi: https://doi.org/10.1039/D0QO01574A

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87. Twofold Radical-Based Synthesis of N,C-Difunctionalized Bicyclo[1.1.1]pentanes

 

H. D. Pickford, J. Nugent, B. Owen, J. J. Mousseau, R. C. Smith and 

E.A. Anderson*

 

J. Am. Chem. Soc.2021143, 9729–9736,

doi: https://doi.org/10.1021/jacs.1c04180

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86. Au(I)-Catalyzed Oxidative Functionalization of Yndiamides

 

Z. Tong, O. L. Garry, P. J. Smith, Y. Jiang, S. J. Mansfield and E. A. Anderson*

 

Org. Lett.2021, 23, 4888–4892,

doi: https://doi.org/10.1021/acs.orglett.1c01625

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85. Synthesis of 1,3-Disubstituted Bicyclo[1.1.0]butanes via Directed Bridgehead Functionalization

 

R. McNamee, M. M. Haugland, J. Nugent, R. Chan, K. Christensen and E. A. Anderson*

 

Chem. Sci.2021, 127480–7485,

doi: https://doi.org/10.1039/D1SC01836A

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84. Marine alkaloids as bioactive agents against protozoal neglected tropical diseases and malaria

 

A. G. Tempone,* P. Pieper, S. E. T. Borborema, F. Thevenard, J. H. G. Lago, S. L. Croft,* E. A. Anderson*

 

Nat. Prod. Rep.2021, Advance Article,

doi: https://doi.org/10.1039/D0NP00078G

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83. Direct catalytic asymmetric synthesis of α-chiral bicyclo[1.1.1]pentanes

 

M. L. J. Wong, A. J. Sterling, J. J. Mousseau, F. Duarte,* E. A. Anderson*

 

Nat. Commun.2021, 12, 1644,

doi: https://doi.org/10.1038/s41467-021-21936-4

Blog post: https://go.nature.com/3uWge10

Highlighted in SYNFORM: 10.1055/s-0040-1720531

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82. Advances in polycyclization cascades in natural product synthesis

 

Y. Jiang,‡ R. E. McNamee,‡ P. J. Smith,‡ A. Sozanschi,‡ Z. Tong,‡ 

E. A. Anderson*

 

Chem. Soc. Rev., 2021, 50, 58–71 doi: https://doi.org/10.1039/D0CS00768D

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81. Synthesis and Structure–Activity Relationship of Dehydrodieugenol B Neolignans against Trypanosoma cruzi

 

C. E. Sear, P. Pieper, M. Amaral, M. M. Romanelli, T. A. Costa-Silva, M. M. Haugland, J. A. Tate, J. H. G. Lago, A. G. Tempone*, E. A. Anderson*

 

ACS Infect. Dis., 2020, 6, 2872–2878, doi: 10.1021/acsinfecdis.0c00523

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80. Site-Selective C–H Benzylation of Alkanes with N-Triftosylhydrazones Leading to Alkyl Aromatics

 

Z. Liu, S. Cao, W. Yu, J. Wu, F. Yi, E. A. Anderson*, X. Bi*

 

Chem, 2020, 6, 2110–2124, doi: 10.1016/j.chempr.2020.06.031

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79. Copper-Catalyzed Intramolecular C–H Alkoxylation of Diaryltriazoles: Synthesis of Tricyclic Triazole Benzoxazines

 

X. Ma, H. Li, H. Xin, W. Du, E. A. Anderson*, X. Dong*, Y. Jiang*

 

Org. Lett., 2020, 22, 5320–5325 doi: 10.1021/acs.orglett.0c01517

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78. Structure-activity relationship study of cytotoxic neolignan derivatives using multivariate analysis and computation-aided drug design

 

F. S. de Sousa, J. L. Baldim, R. A. Azevedo, C. R. Figueiredo, P. Pieper,

C. E. Sear, E. A. Anderson, J. H. G. Lago

 

Bioorg. Med. Chem. Lett., 2020, 30, 127349,

doi: 10.1016/j.bmcl.2020.127349

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77. Synthesis of All-carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron-Catalyzed Kumada Cross-Coupling

 

J. Nugent,‡ B. R. Shire,‡, D. F. J. Caputo, H. D. Pickford, F. Nightingale,

I. T. T. Houlsby, J. J. Mousseau,  E. A. Anderson

equal author contribution

 

Article: Angew. Chem. Int. Ed., 202059, 11866–11870,

            doi: 10.1002/anie.202004090

Featured in: Org. Process Res. Dev., 2020, doi: 10.1021/acs.oprd.0c00344

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76. Rationalizing the diverse reactivity of [1.1.1]propellane through 𝜎-𝜋-delocalization

 

A. J. Sterling, A. B. Dürr, R. C. Smith, E. A. Anderson, F. Duarte

 

Chem. Sci., 2020, 11, 4895–4903. doi: 10.1039/D0SC01386B

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75. 2′-Alkynyl spin-labelling is a minimally perturbing tool for DNA structural analysis

 

J. S. Hardwick, M. M. Haugland, A. H. El-Sagheer, D. Ptchelkine, 

F. R. Beierlein,  A. N. Lane,  T. Brown,  J. E. Lovett,  E. A. Anderson

 

Nucleic Acids Research, 202048, 2830–2840. doi10.1093/nar/gkaa086

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74. A Modular, Enantioselective Synthesis of Resolvins D3, E1, and Hybrids

 

F. Urbitsch, B. L. Elbert, J. Llaveria, P. E. Streatfeild, E. A. Anderson

 

Org. Lett., 202022, 1510–1515. doi: 10.1021/acs.orglett.0c00089

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73. Enantioselective synthesis and anti-parasitic properties of aporphine natural products

 

P. Pieper, E. McHugh, M. Amaral, A. G.Tempone, E. A.Anderson

 

Tetrahedron., 2019, 76, 130814. doi: 10.1016/j.tet.2019.130814

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72. Synthesis of Cyclic Alkenyl Dimethylsiloxanes from Alkynyl Benzyldimethylsilanes and Application in Polyene Synthesis

 

H. G. Gudmundsson, C. J. Kuper, D. Cornut, F. Urbitsch, B. L. Elbert,

E. A. Anderson

 

J. Org. Chem., 201984, 14868-14882. doi: 10.1021/acs.joc.9b01664

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71. Convergent Total Syntheses of (–)-Rubriflordilactone B and (–)-pseudo-Rubriflordilactone B

 

M. Mohammad, V. Chintalapudi, J. M. Carney, S. J. Mansfield, P. Sanderson, K. E. Christensen, E. A. Anderson

 

Angew. Chem. Int. Ed., 201958, 18177–18181. 

doi: 10.1002/anie.201908917

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70. Dehydrodieugenol B derivatives as antiparasitic agents: Synthesis and biological activity against Trypanosoma cruzi

 

D. D. Ferreira, F. S. Sousa, T. A. Costa-Silva, J. Q. Reimão, A. C. Torrecilhas, D. M. Johns, C. E. Sear, K. M. Honorio, J. H. G. Lago, E. A. Anderson, A. G. Tempone

 

Eur. J. Med. Chem.2019, 176, 162-174. doi: 10.1016/j.ejmech.2019.05.001

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69. A semi-synthetic neolignan derivative from dihydrodieugenol B selectively affects the bioenergetic system of Leishmania infantum and inhibits cell division

 

M. Amaral, F. S. de Sousa, T. A. Costa Silva, A. Jimenez G. Junior, N. N. Taniwaki, D. M. Johns, J. H. G. Lago, E. A. Anderson & A. G. Tempone

 

Scientific Reports2019, 6, 6114. doi: 10.1038/s41598-019-42273-z

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68. Silver-Catalyzed C- to N-Center Remote Arene Migration

 

Y. Ning, A. Mekareeya, K. R. Babu, E. A. Anderson and X. Bi

 

ACS Catalysis2019, 9, 4203-4210. doi: 10.1021/acscatal.9b00500

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67. A General Route to Bicyclo[1.1.1]pentanes through Photoredox Catalysis.

 

J. Nugent,* C. Arroniz,* B. R. Shire, A. J. Sterling, H. D. Pickford, M. L. J. Wong,  S. J. Mansfield, D. F. J. Caputo, B. Owen,  J. J. Mousseau, F. Duarte and E. A. Anderson

*equal author contribution

 

ACS Catalysis2019, 9, 9568-9574. doi: 10.1021/acscatal.9b03190

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66. A General Copper-Catalyzed Synthesis of Ynamides from 1,2-Dichloroenamides.

 

S. J. Mansfield, R. C. Smith, J. R. J. Yong, O. L. Garry, and E. A. Anderson

 

Org. Lett., 2019, 21, 2918-2922. doi: 10.1021/acs.orglett.9b00971.

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65. Synthesis of Enantioenriched α-Chiral Bicyclo[1.1.1]pentanes.

 

M. L. J. Wong, J. J. Mousseau, S. J. Mansfield and E. A. Anderson.

 

Org. Lett., 2019, 21, 2408-2411. doi: 10.1021/acs.orglett.9b00691.

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64. Palladium-catalysed ligand-free reductive Heck cycloisomerisation of 1,6-en-α-chloro-enamides. 

 

Y. Hou, J. Ma, H. Yang, E. A. Anderson, A. Whiting and N. Wu. 

 

Chem. Commun., 2019, 55, 3733-3736. doi: 10.1039/C9CC00537D.

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63. Direct Transformation of Terminal Alkynes into Amidines by a Silver-Catalyzed Four-Component Reaction. 

 

B. Liu, Y. Ning, M. Virelli, G. Zanoni, E. A. Anderson and X. Bi. 

 

J. Am. Chem. Soc., 2019, 141, 1593-1598. doi: 10.1021/jacs.8b11039.

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62. Use of trifluoroacetaldehyde N-tfsylhydrazone as a trifluorodiazoethane surrogate and its synthetic applications.

X. Zhang, Z. Liu, X. Yang, Y. Dong, M. Virelli, G. Zanoni, E. A. Anderson and X. Bi. 

 

Nature Commun., 2019, 10, 284doi: 10.1038/s41467-018-08253-z.

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61. Four Step Total Synthesis of an H3 Receptor Antagonist Using Only Tools Found in a Typical Teaching Laboratory.

C. J. Smith, S. J. Mansfield, E. A. Anderson and J. W. Burton. 

 

J. Chem. Educ., 2019, 96, 137-142doi: 10.1021/acs.jchemed.7b00982.